Same Indication

Tofacitinib vs Tofacitinib Citrate

## Tofacitinib vs Tofacitinib Citrate: Overview

This comparison examines the pharmacological differences between **Tofacitinib** and **Tofacitinib Citrate**.

## Mechanism of Action

**Tofacitinib**: Pan-JAK inhibitor with preference for JAK1 and JAK3 blocking pro-inflammatory cytokine signaling.

## Pharmacokinetics

**Half-life**: Tofacitinib — 3.2 hours; Tofacitinib Citrate — N/A.

## Chemical Properties

**Molecular Formula**: Tofacitinib — C16H20N6O; Tofacitinib Citrate — N/A.

**Molecular Weight**: Tofacitinib — 312.3700 g/mol; Tofacitinib Citrate — N/A.

**Type**: Tofacitinib — Small molecule; Tofacitinib Citrate — Small molecule.