Carbamoylcholine

CHEMBL965 Phase 4 معتمد Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
147.2 g/mol
LogP
-0.4
Phase
4

Another name for carbachol, a cholinomimetic agent that activates both muscarinic and nicotinic acetylcholine receptors. It is used as an ophthalmic agent to constrict the pupil and lower intraocular pressure. It is resistant to cholinesterase-mediated breakdown, resulting in a prolonged duration of action.

الوزن الجزيئي

147,2000 g/mol

LogP

-0,40

TPSA

52,30 Ų

قاعدة ليبينسكي للخمسة

ناجح

آلية العمل

Selectively blocks angiotensin II type 1 (AT1) receptors, preventing the vasoconstrictive and aldosterone-secreting effects of angiotensin II. This results in vasodilation, reduced sodium retention, and decreased blood pressure.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

الآلية

Selectively blocks angiotensin II type 1 (AT1) receptors, preventing the vasoconstrictive and aldosterone-secreting effects of angiotensin II. This results in vasodilation, reduced sodium retention, and decreased blood pressure.

البنية ثنائية الأبعاد

SVG PNG

Cite this structure


                        

Embed this structure


                        

SMILES

C[N+](C)(C)CCOC(N)=O

InChI

InChI=1S/C6H14N2O2/c1-8(2,3)4-5-10-6(7)9/h4-5H2,1-3H3,(H-,7,9)/p+1

Molecular Formula

C6H15N2O2+

HBD / HBA

1 / 2

الروابط القابلة للدوران

4

الذرات الثقيلة

10

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

الأسئلة الشائعة

Another name for carbachol, a cholinomimetic agent that activates both muscarinic and nicotinic acetylcholine receptors. It is used as an ophthalmic agent to constrict the pupil and lower intraocular pressure. It is resistant to cholinesterase-mediated breakdown, resulting in a prolonged duration of action.

Selectively blocks angiotensin II type 1 (AT1) receptors, preventing the vasoconstrictive and aldosterone-secreting effects of angiotensin II. This results in vasodilation, reduced sodium retention, and decreased blood pressure.

Yes, Carbamoylcholine is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL965. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 2551. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

إخلاء المسؤولية الطبية

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.