Cenobamate

CHEMBL3989949 Phase 4 معتمد Small molecule

Half-Life

—

Bioavailability

—

Protein Binding

—

Molecular Weight

267.7 g/mol

LogP

1.5

Phase

4

An antiepileptic drug with a dual mechanism, reducing repetitive neuronal firing by blocking sodium channels and enhancing gamma-aminobutyric acid (GABA) activity through modulation of GABAA receptors. It is used as adjunctive therapy for focal-onset seizures in adults. Initiation must be gradual to minimize the risk of a serious multiorgan hypersensitivity reaction called drug reaction with eosinophilia and systemic symptoms (DRESS).

الوزن الجزيئي

267,6700 g/mol

LogP

1,50

TPSA

95,90 Å²

قاعدة ليبينسكي للخمسة

ناجح

المجالات العلاجية

Epilepsy

Pharmacokinetics (PK)

Pharmacodynamics (PD)

البنية ثنائية الأبعاد

SVG PNG

Cite this structure

Embed this structure

SMILES

NC(=O)O[C@@H](Cn1ncnn1)c1ccccc1Cl

InChI

InChI=1S/C10H10ClN5O2/c11-8-4-2-1-3-7(8)9(18-10(12)17)5-16-14-6-13-15-16/h1-4,6,9H,5H2,(H2,12,17)/t9-/m0/s1

Molecular Formula

C10H10ClN5O2

HBD / HBA

1 / 5

الروابط القابلة للدوران

5

الذرات الثقيلة

18

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

الأسئلة الشائعة

An antiepileptic drug with a dual mechanism, reducing repetitive neuronal firing by blocking sodium channels and enhancing gamma-aminobutyric acid (GABA) activity through modulation of GABAA receptors. It is used as adjunctive therapy for focal-onset seizures in adults. Initiation must be gradual to minimize the risk of a serious multiorgan hypersensitivity reaction called drug reaction with eosinophilia and systemic symptoms (DRESS).

Yes, Cenobamate is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

ChEMBL — European Bioinformatics Institute (EBI). CHEMBL3989949. Open-access bioactivity database.
PubChem — National Center for Biotechnology Information (NCBI). CID 11962412. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

PillFYI

هل تبحث عن معلومات ملائمة للمرضى؟

Cenobamate على PillFYI

البنية

بيانات سريعة

الصيغة الجزيئية: C10H10ClN5O2
المرادفات: 1

روابط خارجية

Cite

BibTeX, APA, MLA, Chicago, IEEE, Harvard

إخلاء المسؤولية الطبية

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.