Landiolol

CHEMBL1742466 Phase 4 معتمد Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
509.6 g/mol
LogP
0.1
Phase
4

This ultra-short-acting selective beta-1 blocker is given intravenously to quickly control heart rate in patients with dangerously fast heart rhythms, particularly during or after surgery. Its very brief duration of action allows for precise, rapidly adjustable heart rate control.

الوزن الجزيئي

509,6000 g/mol

LogP

0,10

TPSA

128,00 Ų

قاعدة ليبينسكي للخمسة

ناجح

المجالات العلاجية

Pharmacokinetics (PK)

Pharmacodynamics (PD)

البنية ثنائية الأبعاد

SVG PNG

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SMILES

CC1(C)OC[C@@H](COC(=O)CCc2ccc(OC[C@@H](O)CNCCNC(=O)N3CCOCC3)cc2)O1

InChI

InChI=1S/C25H39N3O8/c1-25(2)35-18-22(36-25)17-34-23(30)8-5-19-3-6-21(7-4-19)33-16-20(29)15-26-9-10-27-24(31)28-11-13-32-14-12-28/h3-4,6-7,20,22,26,29H,5,8-18H2,1-2H3,(H,27,31)/t20-,22+/m0/s1

Molecular Formula

C25H39N3O8

HBD / HBA

3 / 9

الروابط القابلة للدوران

14

الذرات الثقيلة

36

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

الأسئلة الشائعة

This ultra-short-acting selective beta-1 blocker is given intravenously to quickly control heart rate in patients with dangerously fast heart rhythms, particularly during or after surgery. Its very brief duration of action allows for precise, rapidly adjustable heart rate control.

Yes, Landiolol is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1742466. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 114905. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

إخلاء المسؤولية الطبية

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.