Tafenoquine Succinate

CHEMBL2364635 Phase 4 معتمد Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
581.6 g/mol
LogP
Phase
4

Tafenoquine succinate is the succinate salt form of tafenoquine, a long-acting 8-aminoquinoline antimalarial approved for radical cure of Plasmodium vivax malaria and chemoprophylaxis. See tafenoquine for complete pharmacological details.

الوزن الجزيئي

581,6000 g/mol

TPSA

153,00 Ų

المجالات العلاجية

Pharmacokinetics (PK)

Pharmacodynamics (PD)

البنية ثنائية الأبعاد

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SMILES

COc1cc(C)c2c(Oc3cccc(C(F)(F)F)c3)c(OC)cc(NC(C)CCCN)c2n1.O=C(O)CCC(=O)O

InChI

InChI=1S/C24H28F3N3O3.C4H6O4/c1-14-11-20(32-4)30-22-18(29-15(2)7-6-10-28)13-19(31-3)23(21(14)22)33-17-9-5-8-16(12-17)24(25,26)27;5-3(6)1-2-4(7)8/h5,8-9,11-13,15,29H,6-7,10,28H2,1-4H3;1-2H2,(H,5,6)(H,7,8)

Molecular Formula

C28H34F3N3O7

HBD / HBA

4 / 13

الروابط القابلة للدوران

12

الذرات الثقيلة

41

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

الأسئلة الشائعة

Tafenoquine succinate is the succinate salt form of tafenoquine, a long-acting 8-aminoquinoline antimalarial approved for radical cure of Plasmodium vivax malaria and chemoprophylaxis. See tafenoquine for complete pharmacological details.

Yes, Tafenoquine Succinate is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL2364635. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 163761. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

إخلاء المسؤولية الطبية

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.