Betrixaban

CHEMBL512351 Phase 4 Zugelassen Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
451.9 g/mol
LogP
3.6
Phase
4

An oral anticoagulant belonging to the factor Xa inhibitor class, used to prevent blood clots in hospitalized patients at risk for venous thromboembolism. It works by blocking factor Xa, a key enzyme in the blood clotting cascade. Its extended half-life allows for once-daily dosing.

Molekularmasse

451,9000 g/mol

LogP

3,60

TPSA

107,00 Ų

Lipinski-Regel der Fünf

Bestanden

Therapeutische Bereiche

Pharmacokinetics (PK)

Pharmacodynamics (PD)

2D-Struktur

SVG PNG

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SMILES

COc1ccc(NC(=O)c2ccc(C(=N)N(C)C)cc2)c(C(=O)Nc2ccc(Cl)cn2)c1

InChI

InChI=1S/C23H22ClN5O3/c1-29(2)21(25)14-4-6-15(7-5-14)22(30)27-19-10-9-17(32-3)12-18(19)23(31)28-20-11-8-16(24)13-26-20/h4-13,25H,1-3H3,(H,27,30)(H,26,28,31)

Molecular Formula

C23H22ClN5O3

HBD / HBA

3 / 5

Rotierbare Bindungen

7

Schwere Atome

32

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Häufig gestellte Fragen

An oral anticoagulant belonging to the factor Xa inhibitor class, used to prevent blood clots in hospitalized patients at risk for venous thromboembolism. It works by blocking factor Xa, a key enzyme in the blood clotting cascade. Its extended half-life allows for once-daily dosing.

Yes, Betrixaban is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL512351. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 10275777. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

Medizinischer Haftungsausschluss

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.