Difemerine Hydrochloride

CHEMBL3301670 Phase 4 Zugelassen Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
363.9 g/mol
LogP
Phase
4

A hydrochloride salt form of difemerine with the same antispasmodic properties, used to treat gastrointestinal and urinary tract cramping. It works by blocking muscarinic receptors to relax smooth muscle.

Molekularmasse

363,9000 g/mol

TPSA

49,80 Ų

Wirkmechanismus

Competitively blocks muscarinic acetylcholine receptors, reducing parasympathetic nervous system activity. Effects include decreased secretions, bronchodilation, and relaxation of smooth muscle.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Mechanismus

Competitively blocks muscarinic acetylcholine receptors, reducing parasympathetic nervous system activity. Effects include decreased secretions, bronchodilation, and relaxation of smooth muscle.

2D-Struktur

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SMILES

CN(C)CC(C)(C)OC(=O)C(O)(c1ccccc1)c1ccccc1.Cl

InChI

InChI=1S/C20H25NO3.ClH/c1-19(2,15-21(3)4)24-18(22)20(23,16-11-7-5-8-12-16)17-13-9-6-10-14-17;/h5-14,23H,15H2,1-4H3;1H

Molecular Formula

C20H26ClNO3

HBD / HBA

2 / 4

Rotierbare Bindungen

7

Schwere Atome

25

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Häufig gestellte Fragen

A hydrochloride salt form of difemerine with the same antispasmodic properties, used to treat gastrointestinal and urinary tract cramping. It works by blocking muscarinic receptors to relax smooth muscle.

Competitively blocks muscarinic acetylcholine receptors, reducing parasympathetic nervous system activity. Effects include decreased secretions, bronchodilation, and relaxation of smooth muscle.

Yes, Difemerine Hydrochloride is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL3301670. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 3085423. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

Medizinischer Haftungsausschluss

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.