Lidocaine
A local anesthetic and antiarrhythmic used for numbing procedures, nerve blocks, and treating certain heart rhythm abnormalities. It works by blocking sodium channels in nerve and heart muscle cells to prevent electrical signals from propagating.
Molekularmasse
234,3400 g/mol
LogP
2,30
TPSA
32,30 Ų
Lipinski-Regel der Fünf
Bestanden
Therapeutische Bereiche
Wirkmechanismus
Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.
Pharmacokinetics (PK)
Pharmacodynamics (PD)
Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.
2D-Struktur
Cite this structure
Embed this structure
SMILES
CCN(CC)CC(=O)Nc1c(C)cccc1C
InChI
InChI=1S/C14H22N2O/c1-5-16(6-2)10-13(17)15-14-11(3)8-7-9-12(14)4/h7-9H,5-6,10H2,1-4H3,(H,15,17)
Molecular Formula
C14H22N2O
HBD / HBA
1 / 2
Rotierbare Bindungen
5
Schwere Atome
17
No targets recorded
Target interaction data is not yet available for this drug.
No interactions recorded
Drug interaction data is not yet available for this compound.
No side effects recorded
Side effect data is not yet available for this drug.
Häufig gestellte Fragen
A local anesthetic and antiarrhythmic used for numbing procedures, nerve blocks, and treating certain heart rhythm abnormalities. It works by blocking sodium channels in nerve and heart muscle cells to prevent electrical signals from propagating.
Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.
Yes, Lidocaine is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.
References & Data Sources
- ChEMBL — European Bioinformatics Institute (EBI). CHEMBL79. Open-access bioactivity database.
- PubChem — National Center for Biotechnology Information (NCBI). CID 3676. Chemical information database.
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.
Medizinischer Haftungsausschluss
This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.
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