Tetracaine Hydrochloride

CHEMBL1255654 Phase 4 Zugelassen Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
300.8 g/mol
LogP
Phase
4

A hydrochloride salt form of tetracaine with the same therapeutic properties. This local anesthetic is used to numb specific areas of the body before medical procedures, and is commonly used as eye drops before eye examinations or minor eye surgery, as well as in spinal anesthesia.

Molekularmasse

300,8200 g/mol

TPSA

41,60 Ų

Therapeutische Bereiche

Wirkmechanismus

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Mechanismus

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

2D-Struktur

SVG PNG

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SMILES

CCCCNc1ccc(C(=O)OCCN(C)C)cc1.Cl

InChI

InChI=1S/C15H24N2O2.ClH/c1-4-5-10-16-14-8-6-13(7-9-14)15(18)19-12-11-17(2)3;/h6-9,16H,4-5,10-12H2,1-3H3;1H

Molecular Formula

C15H25ClN2O2

HBD / HBA

2 / 4

Rotierbare Bindungen

9

Schwere Atome

20

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Häufig gestellte Fragen

A hydrochloride salt form of tetracaine with the same therapeutic properties. This local anesthetic is used to numb specific areas of the body before medical procedures, and is commonly used as eye drops before eye examinations or minor eye surgery, as well as in spinal anesthesia.

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Yes, Tetracaine Hydrochloride is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1255654. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 8695. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

Medizinischer Haftungsausschluss

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.