Isoetharine Mesylate
This mesylate salt of isoetharine is a short-acting beta-agonist bronchodilator previously used in nebulizer solutions for asthma and bronchospasm relief. It stimulates beta-2 adrenergic receptors to relax airway smooth muscle. Newer selective and longer-acting beta-agonists have largely replaced it in clinical practice.
Peso molecular
335,4200 g/mol
TPSA
135,00 Ų
Mecanismo de acción
Activates beta-2 adrenergic receptors on bronchial smooth muscle, stimulating adenylyl cyclase and increasing intracellular cAMP. This relaxes airway smooth muscle and produces bronchodilation.
Pharmacokinetics (PK)
Pharmacodynamics (PD)
Activates beta-2 adrenergic receptors on bronchial smooth muscle, stimulating adenylyl cyclase and increasing intracellular cAMP. This relaxes airway smooth muscle and produces bronchodilation.
Estructura 2D
Cite this structure
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SMILES
CCC(NC(C)C)C(O)c1ccc(O)c(O)c1.CS(=O)(=O)O
InChI
InChI=1S/C13H21NO3.CH4O3S/c1-4-10(14-8(2)3)13(17)9-5-6-11(15)12(16)7-9;1-5(2,3)4/h5-8,10,13-17H,4H2,1-3H3;1H3,(H,2,3,4)
Molecular Formula
C14H25NO6S
HBD / HBA
5 / 7
Enlaces Rotables
5
Átomos Pesados
22
No targets recorded
Target interaction data is not yet available for this drug.
No interactions recorded
Drug interaction data is not yet available for this compound.
No side effects recorded
Side effect data is not yet available for this drug.
Preguntas frecuentes
This mesylate salt of isoetharine is a short-acting beta-agonist bronchodilator previously used in nebulizer solutions for asthma and bronchospasm relief. It stimulates beta-2 adrenergic receptors to relax airway smooth muscle. Newer selective and longer-acting beta-agonists have largely replaced it in clinical practice.
Activates beta-2 adrenergic receptors on bronchial smooth muscle, stimulating adenylyl cyclase and increasing intracellular cAMP. This relaxes airway smooth muscle and produces bronchodilation.
Yes, Isoetharine Mesylate is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.
References & Data Sources
- ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1201153. Open-access bioactivity database.
- PubChem — National Center for Biotechnology Information (NCBI). CID 23702. Chemical information database.
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.
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