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Lidocaine Hydrochloride

CHEMBL1200409 Phase 4 Aprobado Small molecule
Half-Life
—
Bioavailability
—
Protein Binding
—
Molecular Weight
270.8 g/mol
LogP
—
Phase
4

The hydrochloride salt form of lidocaine, the most commonly used preparation for local anesthesia and intravenous antiarrhythmic therapy. It is used in everything from dental procedures to treating life-threatening arrhythmias.

Peso molecular

270,8000 g/mol

TPSA

32,30 Ų

Áreas terapéuticas

Anestesiología Artritis reumatoide Asma Cáncer colorrectal Cáncer de mama Cáncer de ovario Cáncer de páncreas Cáncer de próstata Cáncer de pulmón de células no pequeñas Cáncer de tiroides Cáncer de vejiga Degeneración macular relacionada con la edad Dermatitis atópica Dermatología Diabetes tipo 2 Dolor crónico Endocrinología Endometriosis Enfermedad cardiovascular Enfermedad de Alzheimer Enfermedad del hígado graso no alcohólico Enfermedad de Parkinson Enfermedad infecciosa Enfermedad inflamatoria intestinal Enfermedad por reflujo gastroesofágico Enfermedad pulmonar obstructiva crónica Enfermedad renal crónica Enfermedad respiratoria Epilepsia Esclerosis múltiple Esquizofrenia Fibrilación auricular Gastroenterología Glaucoma Gota Hematología Hepatitis C Hepatología Hiperlipidemia Hiperplasia prostática benigna Hipertensión Ictus Inmunología Insomnio Insuficiencia cardíaca Leucemia Linfoma Lupus eritematoso sistémico Malaria Manejo del dolor Medicina de trasplantes Melanoma Migraña Nefrología Neurología Obesidad Obstetricia y ginecología Oftalmología Oncología Osteoporosis Psiquiatría Psoriasis Reumatología Trastorno bipolar Trastorno de ansiedad generalizada Trastorno depresivo mayor Trombosis venosa profunda / Embolia pulmonar Tuberculosis Urología VIH/sida

Mecanismo de acción

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Mecanismo

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Estructura 2D

SVG PNG

Cite this structure


                        

                            
                            
                        

                    

                


                
                

                    

                    

                        
Embed this structure

                        

                        

                            
                            
                        

                    

                

                

                
                

                    
SMILES

                    
CCN(CC)CC(=O)Nc1c(C)cccc1C.Cl.O

                

                

                
                

                    
InChI

                    
InChI=1S/C14H22N2O.ClH.H2O/c1-5-16(6-2)10-13(17)15-14-11(3)8-7-9-12(14)4;;/h7-9H,5-6,10H2,1-4H3,(H,15,17);1H;1H2

                

                

                

                    
                    

                        
Molecular Formula

                        
C14H23ClN2O

                    

                    
                    

                        
HBD / HBA

                        
2 / 2

                    

                    
                    

                        
Enlaces Rotables

                        
5

                    

                    
                    
                    

                        
Átomos Pesados

                        
18

                    

                    
                

            


            
            

                
                


    
    
        
    
    
    
No targets recorded

    
    
Target interaction data is not yet available for this drug.

    



                
            


            
            

                
                


    
    
        
    
    
    
No interactions recorded

    
    
Drug interaction data is not yet available for this compound.

    



                
            


            
            

                
                


    
    
        
    
    
    
No side effects recorded

    
    
Side effect data is not yet available for this drug.

    



                
            


            
            
            

                
Preguntas frecuentes

                

                    
                    

                        
                        

                            
The hydrochloride salt form of lidocaine, the most commonly used preparation for local anesthesia and intravenous antiarrhythmic therapy. It is used in everything from dental procedures to treating life-threatening arrhythmias.

                        

                    

                    

                    

                    
                    

                        
                        

                            
Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

                        

                    

                    

                    

                    

                        
                        

                            
Yes, Lidocaine Hydrochloride is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

                        

                    

                

            

            

            
            

            
            

            
            
{# References & Data Sources section for drug detail pages.
   Renders standard pharmacological database links plus the drug's data_sources field. #}


    
References & Data Sources

    
    
        
        
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                ChEMBL — European Bioinformatics Institute (EBI).
                CHEMBL1200409.
                Open-access bioactivity database.
            
        
    • 
        
        
        
  • 
            
            
                PubChem — National Center for Biotechnology Information (NCBI).
                CID 6314.
                Chemical information database.
            
        
    • 
        
        
        
        
    

    
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.




        


        
        
    


    



    
Aviso médico

    

        This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.
    

    

        Data sources:
        ChEMBL,
        PubChem,
        DailyMed.