Diazoxide

CHEMBL181 Phase 4 Approuvé Small molecule

Half-Life

—

Bioavailability

—

Protein Binding

—

Molecular Weight

230.7 g/mol

LogP

1.2

Phase

4

A potassium channel opener that lowers blood sugar by inhibiting insulin secretion from the pancreas, used to treat persistent hypoglycemia from hyperinsulinism, and formerly used intravenously for hypertensive emergencies. Oral diazoxide is now primarily used for congenital hyperinsulinism.

Masse moléculaire

230,6700 g/mol

LogP

1,20

TPSA

66,90 Å²

Règle des 5 de Lipinski

Conforme

Aires thérapeutiques

Ovarian Cancer Non-Alcoholic Fatty Liver Disease Obesity Type 2 Diabetes

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Structure 2D

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SMILES

CC1=Nc2ccc(Cl)cc2S(=O)(=O)N1

InChI

InChI=1S/C8H7ClN2O2S/c1-5-10-7-3-2-6(9)4-8(7)14(12,13)11-5/h2-4H,1H3,(H,10,11)

Molecular Formula

C8H7ClN2O2S

HBD / HBA

1 / 3

Liaisons Rotatives

0

Atomes Lourds

14

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Foire aux questions

A potassium channel opener that lowers blood sugar by inhibiting insulin secretion from the pancreas, used to treat persistent hypoglycemia from hyperinsulinism, and formerly used intravenously for hypertensive emergencies. Oral diazoxide is now primarily used for congenital hyperinsulinism.

Yes, Diazoxide is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

ChEMBL — European Bioinformatics Institute (EBI). CHEMBL181. Open-access bioactivity database.
PubChem — National Center for Biotechnology Information (NCBI). CID 3019. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

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Structure

Données Clés

Formule: C8H7ClN2O2S
Synonymes: 3

Liens externes

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Avertissement médical

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.