Cisapride Monohydrate

CHEMBL1200788 Phase 4 Disetujui Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
484.0 g/mol
LogP
Phase
4

The monohydrate form of cisapride was the standard clinical formulation of this gastroprokinetic agent. It shares the same efficacy and the same serious cardiac arrhythmia risk as the parent compound. Its withdrawal from most markets due to fatal QT prolongation represents a landmark in drug safety.

Berat Molekul

484,0000 g/mol

TPSA

87,10 Ų

Area Terapeutik

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Struktur 2D

SVG PNG

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SMILES

COc1cc(N)c(Cl)cc1C(=O)NC1CCN(CCCOc2ccc(F)cc2)CC1OC.O

InChI

InChI=1S/C23H29ClFN3O4.H2O/c1-30-21-13-19(26)18(24)12-17(21)23(29)27-20-8-10-28(14-22(20)31-2)9-3-11-32-16-6-4-15(25)5-7-16;/h4-7,12-13,20,22H,3,8-11,14,26H2,1-2H3,(H,27,29);1H2

Molecular Formula

C23H31ClFN3O5

HBD / HBA

3 / 8

Ikatan yang Dapat Dirotasi

9

Atom Berat

33

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Pertanyaan yang Sering Diajukan

The monohydrate form of cisapride was the standard clinical formulation of this gastroprokinetic agent. It shares the same efficacy and the same serious cardiac arrhythmia risk as the parent compound. Its withdrawal from most markets due to fatal QT prolongation represents a landmark in drug safety.

Yes, Cisapride Monohydrate is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1200788. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 6917697. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

Penyangkalan Medis

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.