Gallium Ga 68 Gozetotide

CHEMBL5095039 Phase 4 Disetujui Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
1011.9 g/mol
LogP
Phase
4

This radioactive diagnostic agent is used in PET imaging to detect prostate cancer that has spread or recurred. It binds to prostate-specific membrane antigen (PSMA), a protein highly expressed on prostate cancer cells, allowing the imaging device to locate even small deposits of cancer. It is particularly useful when conventional imaging may not detect disease recurrence.

Berat Molekul

1011,9000 g/mol

TPSA

381,00 Ų

Area Terapeutik

Mekanisme Kerja

Functions as a diagnostic agent by providing contrast enhancement or radioactive tracer activity that enables visualization of anatomical structures or physiological processes during medical imaging.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Mekanisme

Functions as a diagnostic agent by providing contrast enhancement or radioactive tracer activity that enables visualization of anatomical structures or physiological processes during medical imaging.

Struktur 2D

SVG PNG

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SMILES

O=C([O-])CN(CCN(CC(=O)[O-])Cc1cc(CCC(=O)NCCCCCC(=O)NCCCC[C@H](NC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O)ccc1[O-])Cc1cc(CCC(=O)O)ccc1[O-].[68Ga+3].[OH3+]

InChI

InChI=1S/C44H62N6O17.Ga.H2O/c51-34-13-8-28(22-30(34)24-49(26-40(59)60)20-21-50(27-41(61)62)25-31-23-29(9-14-35(31)52)11-16-38(55)56)10-15-37(54)46-18-4-1-2-7-36(53)45-19-5-3-6-32(42(63)64)47-44(67)48-33(43(65)66)12-17-39(57)58;;/h8-9,13-14,22-23,32-33,51-52H,1-7,10-12,15-21,24-27H2,(H,45,53)(H,46,54)(H,55,56)(H,57,58)(H,59,60)(H,61,62)(H,63,64)(H,65,66)(H2,47,48,67);;1H2/q;+3;/p-3/t32-,33-;;/m0../s1/i;1-2;

Molecular Formula

C44H59GaN6O17

HBD / HBA

9 / 19

Ikatan yang Dapat Dirotasi

33

Atom Berat

68

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Pertanyaan yang Sering Diajukan

This radioactive diagnostic agent is used in PET imaging to detect prostate cancer that has spread or recurred. It binds to prostate-specific membrane antigen (PSMA), a protein highly expressed on prostate cancer cells, allowing the imaging device to locate even small deposits of cancer. It is particularly useful when conventional imaging may not detect disease recurrence.

Functions as a diagnostic agent by providing contrast enhancement or radioactive tracer activity that enables visualization of anatomical structures or physiological processes during medical imaging.

Yes, Gallium Ga 68 Gozetotide is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL5095039. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 154572876. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

Penyangkalan Medis

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.