Timolol

CHEMBL499 Phase 4 Disetujui Small molecule

Half-Life

—

Bioavailability

—

Protein Binding

—

Molecular Weight

316.4 g/mol

LogP

1.8

Phase

4

This beta-blocker medication is used to lower high blood pressure, prevent migraine headaches, reduce the risk of further heart attacks, and — most commonly as eye drops — to lower elevated eye pressure in glaucoma and ocular hypertension. It works by blocking adrenaline-like signals that would otherwise speed up the heart and constrict blood vessels. As eye drops, it can still be absorbed into the bloodstream and affect heart rate in sensitive individuals.

Berat Molekul

316,4200 g/mol

LogP

1,80

TPSA

108,00 Å²

Lipinski RO5

Lulus

Area Terapeutik

Melanoma Glaucoma Age-Related Macular Degeneration Migraine Hypertension

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Struktur 2D

SVG PNG

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SMILES

CC(C)(C)NC[C@H](O)COc1nsnc1N1CCOCC1

InChI

InChI=1S/C13H24N4O3S/c1-13(2,3)14-8-10(18)9-20-12-11(15-21-16-12)17-4-6-19-7-5-17/h10,14,18H,4-9H2,1-3H3/t10-/m0/s1

Molecular Formula

C13H24N4O3S

HBD / HBA

2 / 8

Ikatan yang Dapat Dirotasi

7

Atom Berat

21

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Pertanyaan yang Sering Diajukan

This beta-blocker medication is used to lower high blood pressure, prevent migraine headaches, reduce the risk of further heart attacks, and — most commonly as eye drops — to lower elevated eye pressure in glaucoma and ocular hypertension. It works by blocking adrenaline-like signals that would otherwise speed up the heart and constrict blood vessels. As eye drops, it can still be absorbed into the bloodstream and affect heart rate in sensitive individuals.

Yes, Timolol is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

ChEMBL — European Bioinformatics Institute (EBI). CHEMBL499. Open-access bioactivity database.
PubChem — National Center for Biotechnology Information (NCBI). CID 33624. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

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Struktur

Data Cepat

Rumus: C13H24N4O3S
Sinonim: 24

Tautan Eksternal

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Penyangkalan Medis

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.