Major Established

Deskripsi

Dual RAAS blockade with ACE inhibitors and ARBs provides no additional cardiovascular benefit over either agent alone and significantly increases the risk of hypotension, hyperkalemia, and acute kidney injury.

Mekanisme

Both drugs block angiotensin II effects (ACEi prevents its synthesis; ARB blocks AT1 receptors); combination results in excessive RAAS inhibition, causing additive hypotension, reduced aldosterone (hyperkalemia), and impaired renal autoregulation.

Signifikansi Klinis

ONTARGET trial demonstrated no cardiovascular benefit with dual blockade but significantly higher rates of hypotension (4.8%), syncope, diarrhea, renal impairment, and hyperkalemia.

Penatalaksanaan

Avoid dual RAAS blockade in most patients. Exception: select cases of refractory heart failure under specialist supervision with close monitoring of BP, renal function, and potassium.

Penyangkalan Medis

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.