PPARG (Peroxisome Proliferator-Activated Receptor Gamma)
PPARG
Nuclear receptor regulating glucose and lipid metabolism, adipocyte differentiation.
Fungsi
Thiazolidinediones (pioglitazone) activate PPARG to improve insulin sensitivity.
Obat yang Bekerja pada Target Ini
| Obat | Aksi | Utama |
|---|---|---|
| Methylprednisolone | Agonist | Ya |
| Insulin Glargine | Agonist | Ya |
| Liraglutide | Agonist | Ya |
| Semaglutide | Agonist | Ya |
| Tirzepatide | Agonist | Ya |
| Prednisone | Agonist | Ya |
| Dexamethasone | Agonist | Ya |
| Levothyroxine | Agonist | Ya |
| Spironolactone | Antagonist | Ya |
| Tamoxifen | Antagonist | Ya |
| Sitagliptin | Inhibitor | Ya |
| Finasteride | Inhibitor | Ya |
| Empagliflozin | Inhibitor | Ya |
| Metformin | Other | Ya |
| Montelukast | Other | — |