Etidocaine

CHEMBL492 Phase 4 承認済み Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
276.4 g/mol
LogP
3.7
Phase
4

This local anesthetic blocks sodium channels in nerve cells to prevent pain signals from being transmitted during surgical procedures or dental work. It provides profound motor and sensory blockade.

分子量

276.4000 g/mol

LogP

3.70

TPSA

32.30 Ų

リピンスキーの五則

適合

作用機序

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

機序

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

2D構造

SVG PNG

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SMILES

CCCN(CC)C(CC)C(=O)Nc1c(C)cccc1C

InChI

InChI=1S/C17H28N2O/c1-6-12-19(8-3)15(7-2)17(20)18-16-13(4)10-9-11-14(16)5/h9-11,15H,6-8,12H2,1-5H3,(H,18,20)

Molecular Formula

C17H28N2O

HBD / HBA

1 / 2

回転可能結合数

7

重原子数

20

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

よくある質問

This local anesthetic blocks sodium channels in nerve cells to prevent pain signals from being transmitted during surgical procedures or dental work. It provides profound motor and sensory blockade.

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Yes, Etidocaine is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL492. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 37497. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

医学的免責事項

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.