Halazepam

CHEMBL970 Phase 4 承認済み Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
352.7 g/mol
LogP
4.0
Phase
4

This benzodiazepine medication acts on the central nervous system to produce anxiolytic, sedative, muscle relaxant, and anticonvulsant effects. It was used to treat anxiety disorders but has been withdrawn from the market in some countries. Like all benzodiazepines, it carries a risk of dependence and withdrawal symptoms with prolonged use.

分子量

352.7000 g/mol

LogP

4.00

TPSA

32.70 Ų

リピンスキーの五則

適合

作用機序

Reduces skeletal muscle tone and spasm through central or peripheral mechanisms, typically by modulating spinal reflexes, enhancing inhibitory neurotransmission, or blocking neuromuscular transmission.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

機序

Reduces skeletal muscle tone and spasm through central or peripheral mechanisms, typically by modulating spinal reflexes, enhancing inhibitory neurotransmission, or blocking neuromuscular transmission.

2D構造

SVG PNG

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SMILES

O=C1CN=C(c2ccccc2)c2cc(Cl)ccc2N1CC(F)(F)F

InChI

InChI=1S/C17H12ClF3N2O/c18-12-6-7-14-13(8-12)16(11-4-2-1-3-5-11)22-9-15(24)23(14)10-17(19,20)21/h1-8H,9-10H2

Molecular Formula

C17H12ClF3N2O

HBD / HBA

- / 5

回転可能結合数

2

重原子数

24

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

よくある質問

This benzodiazepine medication acts on the central nervous system to produce anxiolytic, sedative, muscle relaxant, and anticonvulsant effects. It was used to treat anxiety disorders but has been withdrawn from the market in some countries. Like all benzodiazepines, it carries a risk of dependence and withdrawal symptoms with prolonged use.

Reduces skeletal muscle tone and spasm through central or peripheral mechanisms, typically by modulating spinal reflexes, enhancing inhibitory neurotransmission, or blocking neuromuscular transmission.

Yes, Halazepam is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL970. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 31640. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

医学的免責事項

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.