Pyrovalerone
Pyrovalerone is a psychostimulant cathinone derivative that inhibits the reuptake of dopamine and norepinephrine by blocking their respective monoamine transporters, producing CNS stimulation, increased alertness, and euphoria similar to cocaine. It was briefly investigated as a treatment for fatigue and lethargy but is now a controlled substance due to its significant abuse potential.
分子量
245.3600 g/mol
LogP
3.80
TPSA
20.30 Ų
リピンスキーの五則
適合
Pharmacokinetics (PK)
Pharmacodynamics (PD)
2D構造
Cite this structure
Embed this structure
SMILES
CCCC(C(=O)c1ccc(C)cc1)N1CCCC1
InChI
InChI=1S/C16H23NO/c1-3-6-15(17-11-4-5-12-17)16(18)14-9-7-13(2)8-10-14/h7-10,15H,3-6,11-12H2,1-2H3
Molecular Formula
C16H23NO
HBD / HBA
- / 2
回転可能結合数
5
重原子数
18
No targets recorded
Target interaction data is not yet available for this drug.
No interactions recorded
Drug interaction data is not yet available for this compound.
No side effects recorded
Side effect data is not yet available for this drug.
よくある質問
Pyrovalerone is a psychostimulant cathinone derivative that inhibits the reuptake of dopamine and norepinephrine by blocking their respective monoamine transporters, producing CNS stimulation, increased alertness, and euphoria similar to cocaine. It was briefly investigated as a treatment for fatigue and lethargy but is now a controlled substance due to its significant abuse potential.
Yes, Pyrovalerone is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.
References & Data Sources
- ChEMBL — European Bioinformatics Institute (EBI). CHEMBL201960. Open-access bioactivity database.
- PubChem — National Center for Biotechnology Information (NCBI). CID 14373. Chemical information database.
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.
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