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Selexipag

CHEMBL238804 Phase 4 承認済み Small molecule
Half-Life
—
Bioavailability
—
Protein Binding
—
Molecular Weight
496.6 g/mol
LogP
3.8
Phase
4

Taken orally twice daily, this medication mimics the action of a natural substance called prostacyclin to relax and widen the blood vessels in the lungs, reducing the pressure that the heart must work against. It helps slow the progression of pulmonary arterial hypertension and lowers the risk of disease worsening requiring hospitalization.

分子量

496.6000 g/mol

LogP

3.80

TPSA

110.00 Ų

リピンスキーの五則

適合

治療領域

Hypertension

Pharmacokinetics (PK)

Pharmacodynamics (PD)

2D構造

SVG PNG

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SMILES

                    
CC(C)N(CCCCOCC(=O)NS(C)(=O)=O)c1cnc(-c2ccccc2)c(-c2ccccc2)n1

                

                

                
                

                    
InChI

                    
InChI=1S/C26H32N4O4S/c1-20(2)30(16-10-11-17-34-19-24(31)29-35(3,32)33)23-18-27-25(21-12-6-4-7-13-21)26(28-23)22-14-8-5-9-15-22/h4-9,12-15,18,20H,10-11,16-17,19H2,1-3H3,(H,29,31)

                

                

                

                    
                    

                        
Molecular Formula

                        
C26H32N4O4S

                    

                    
                    

                        
HBD / HBA

                        
1 / 7

                    

                    
                    

                        
回転可能結合数

                        
12

                    

                    
                    
                    

                        
重原子数

                        
35

                    

                    
                

            


            
            

                
                


    
    
        
    
    
    
No targets recorded

    
    
Target interaction data is not yet available for this drug.

    



                
            


            
            

                
                


    
    
        
    
    
    
No interactions recorded

    
    
Drug interaction data is not yet available for this compound.

    



                
            


            
            

                
                


    
    
        
    
    
    
No side effects recorded

    
    
Side effect data is not yet available for this drug.

    



                
            


            
            
            

                
よくある質問

                

                    
                    

                        
                        

                            
Taken orally twice daily, this medication mimics the action of a natural substance called prostacyclin to relax and widen the blood vessels in the lungs, reducing the pressure that the heart must work against. It helps slow the progression of pulmonary arterial hypertension and lowers the risk of disease worsening requiring hospitalization.

                        

                    

                    

                    

                    

                    

                    

                        
                        

                            
Yes, Selexipag is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

                        

                    

                

            

            

            
            

            
            

            
            
{# References & Data Sources section for drug detail pages.
   Renders standard pharmacological database links plus the drug's data_sources field. #}


    
References & Data Sources

    
    
        
        
  • 
            
            
                ChEMBL — European Bioinformatics Institute (EBI).
                CHEMBL238804.
                Open-access bioactivity database.
            
        
    • 
        
        
        
  • 
            
            
                PubChem — National Center for Biotechnology Information (NCBI).
                CID 9913767.
                Chemical information database.
            
        
    • 
        
        
        
        
    

    
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.




        


        
        
    


    



    
医学的免責事項

    

        This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.
    

    

        Data sources:
        ChEMBL,
        PubChem,
        DailyMed.