PPARG (Peroxisome Proliferator-Activated Receptor Gamma)
PPARG
Nuclear receptor regulating glucose and lipid metabolism, adipocyte differentiation.
機能
Thiazolidinediones (pioglitazone) activate PPARG to improve insulin sensitivity.
この標的に作用する薬物
| 薬物 | 作用 | 主要 |
|---|---|---|
| Methylprednisolone | Agonist | はい |
| Insulin Glargine | Agonist | はい |
| Liraglutide | Agonist | はい |
| Semaglutide | Agonist | はい |
| Tirzepatide | Agonist | はい |
| Prednisone | Agonist | はい |
| Dexamethasone | Agonist | はい |
| Levothyroxine | Agonist | はい |
| Spironolactone | Antagonist | はい |
| Tamoxifen | Antagonist | はい |
| Sitagliptin | Inhibitor | はい |
| Finasteride | Inhibitor | はい |
| Empagliflozin | Inhibitor | はい |
| Metformin | Other | はい |
| Montelukast | Other | — |