Bremelanotide Acetate

CHEMBL4297533 Phase 4 승인됨 Protein
Half-Life
Bioavailability
Protein Binding
Molecular Weight
1085.2 g/mol
LogP
Phase
4

The acetate salt form of bremelanotide, approved to treat acquired generalized hypoactive sexual desire disorder in premenopausal women. It stimulates melanocortin receptors in the central nervous system to enhance sexual desire. Nausea and temporary increases in blood pressure are among its notable side effects.

분자량

1085.2000 g/mol

TPSA

416.00 Ų

치료 영역

작용 기전

Binds to and activates its target receptor, mimicking the action of the endogenous ligand to produce a specific physiological response.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

기전

Binds to and activates its target receptor, mimicking the action of the endogenous ligand to produce a specific physiological response.

2D 구조

SVG PNG

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SMILES

CC(=O)O.CCCC[C@H](NC(C)=O)C(=O)N[C@H]1CC(=O)NCCCC[C@@H](C(=O)O)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]cn2)NC1=O

InChI

InChI=1S/C50H68N14O10.C2H4O2/c1-3-4-16-35(58-29(2)65)43(67)64-41-25-42(66)54-20-11-10-18-37(49(73)74)60-46(70)39(23-31-26-56-34-17-9-8-15-33(31)34)62-44(68)36(19-12-21-55-50(51)52)59-45(69)38(22-30-13-6-5-7-14-30)61-47(71)40(63-48(41)72)24-32-27-53-28-57-32;1-2(3)4/h5-9,13-15,17,26-28,35-41,56H,3-4,10-12,16,18-25H2,1-2H3,(H,53,57)(H,54,66)(H,58,65)(H,59,69)(H,60,70)(H,61,71)(H,62,68)(H,63,72)(H,64,67)(H,73,74)(H4,51,52,55);1H3,(H,3,4)/t35-,36-,37-,38+,39-,40-,41-;/m0./s1

Molecular Formula

C52H72N14O12

HBD / HBA

14 / 14

회전 가능 결합

17

무거운 원자

78

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

자주 묻는 질문

The acetate salt form of bremelanotide, approved to treat acquired generalized hypoactive sexual desire disorder in premenopausal women. It stimulates melanocortin receptors in the central nervous system to enhance sexual desire. Nausea and temporary increases in blood pressure are among its notable side effects.

Binds to and activates its target receptor, mimicking the action of the endogenous ligand to produce a specific physiological response.

Yes, Bremelanotide Acetate is an approved drug. It has reached clinical phase 4. It is classified as a Protein.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL4297533. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 91971505. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

의학적 면책조항

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.