Tamoxifen Citrate

CHEMBL786 Phase 4 승인됨 Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
563.6 g/mol
LogP
Phase
4

A citrate salt form of tamoxifen with the same therapeutic properties. This medication blocks estrogen receptors in breast tissue and is widely used to treat and reduce the risk of hormone receptor-positive breast cancer in both women and men.

분자량

563.6000 g/mol

TPSA

145.00 Ų

치료 영역

작용 기전

Selective estrogen receptor modulator (SERM).

Pharmacokinetics (PK)

Pharmacodynamics (PD)

기전

Selective estrogen receptor modulator (SERM).

2D 구조

SVG PNG

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SMILES

CC/C(=C(\c1ccccc1)c1ccc(OCCN(C)C)cc1)c1ccccc1.O=C(O)CC(O)(CC(=O)O)C(=O)O

InChI

InChI=1S/C26H29NO.C6H8O7/c1-4-25(21-11-7-5-8-12-21)26(22-13-9-6-10-14-22)23-15-17-24(18-16-23)28-20-19-27(2)3;7-3(8)1-6(13,5(11)12)2-4(9)10/h5-18H,4,19-20H2,1-3H3;13H,1-2H2,(H,7,8)(H,9,10)(H,11,12)/b26-25-;

Molecular Formula

C32H37NO8

HBD / HBA

4 / 9

회전 가능 결합

13

무거운 원자

41

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

자주 묻는 질문

A citrate salt form of tamoxifen with the same therapeutic properties. This medication blocks estrogen receptors in breast tissue and is widely used to treat and reduce the risk of hormone receptor-positive breast cancer in both women and men.

Selective estrogen receptor modulator (SERM).

Yes, Tamoxifen Citrate is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL786. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 2733525. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

의학적 면책조항

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.