Moderate Established

설명

Combining adalimumab with cyclosporine produces substantial additive immunosuppression, increasing the risk of serious opportunistic infections, lymphoma, and other immunosuppression-related malignancies.

기전

Adalimumab blocks TNF-alpha, impairing macrophage-dependent defence against intracellular pathogens; cyclosporine inhibits T-cell activation via calcineurin inhibition, further blunting adaptive immunity. The combination suppresses both innate and adaptive immune responses.

임상적 중요성

Post-marketing data and registry studies report markedly elevated rates of serious infections (tuberculosis reactivation, invasive fungal infections, PML) with biologic + CNI combinations.

관리 방법

Avoid combination unless a compelling clinical indication exists; screen for latent tuberculosis and hepatitis B before initiating; monitor for signs of infection; do not administer live vaccines during therapy.

의학적 면책조항

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.