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Bexarotene

CHEMBL1023 Phase 4 Одобрено Small molecule
Half-Life
—
Bioavailability
—
Protein Binding
—
Molecular Weight
348.5 g/mol
LogP
7.6
Phase
4

A retinoid medication that activates a specific class of receptors called retinoid X receptors to regulate cell growth and differentiation. It is used to treat cutaneous T-cell lymphoma, a rare cancer affecting the skin. Side effects include elevated lipid levels and serious thyroid abnormalities requiring close monitoring.

Молекулярная масса

348,5000 g/mol

LogP

7,60

TPSA

37,30 Ų

Правило пяти Липинского

Соответствует

Терапевтические области

Thyroid Cancer Non-Small Cell Lung Cancer Alzheimer's Disease Schizophrenia Psoriasis Lymphoma Breast Cancer Leukemia

Pharmacokinetics (PK)

Pharmacodynamics (PD)

2D Структура

SVG PNG

Cite this structure


                        

                            
                            
                        

                    

                


                
                

                    

                    

                        
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SMILES

                    
C=C(c1ccc(C(=O)O)cc1)c1cc2c(cc1C)C(C)(C)CCC2(C)C

                

                

                
                

                    
InChI

                    
InChI=1S/C24H28O2/c1-15-13-20-21(24(5,6)12-11-23(20,3)4)14-19(15)16(2)17-7-9-18(10-8-17)22(25)26/h7-10,13-14H,2,11-12H2,1,3-6H3,(H,25,26)

                

                

                

                    
                    

                        
Molecular Formula

                        
C24H28O2

                    

                    
                    

                        
HBD / HBA

                        
1 / 2

                    

                    
                    

                        
Вращаемые Связи

                        
3

                    

                    
                    
                    

                        
Тяжёлые Атомы

                        
26

                    

                    
                

            


            
            

                
                


    
    
        
    
    
    
No targets recorded

    
    
Target interaction data is not yet available for this drug.

    



                
            


            
            

                
                


    
    
        
    
    
    
No interactions recorded

    
    
Drug interaction data is not yet available for this compound.

    



                
            


            
            

                
                


    
    
        
    
    
    
No side effects recorded

    
    
Side effect data is not yet available for this drug.

    



                
            


            
            
            

                
Часто задаваемые вопросы

                

                    
                    

                        
                        

                            
A retinoid medication that activates a specific class of receptors called retinoid X receptors to regulate cell growth and differentiation. It is used to treat cutaneous T-cell lymphoma, a rare cancer affecting the skin. Side effects include elevated lipid levels and serious thyroid abnormalities requiring close monitoring.

                        

                    

                    

                    

                    

                    

                    

                        
                        

                            
Yes, Bexarotene is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

                        

                    

                

            

            

            
            

            
            

            
            
{# References & Data Sources section for drug detail pages.
   Renders standard pharmacological database links plus the drug's data_sources field. #}


    
References & Data Sources

    
    
        
        
  • 
            
            
                ChEMBL — European Bioinformatics Institute (EBI).
                CHEMBL1023.
                Open-access bioactivity database.
            
        
    • 
        
        
        
  • 
            
            
                PubChem — National Center for Biotechnology Information (NCBI).
                CID 82146.
                Chemical information database.
            
        
    • 
        
        
        
        
    

    
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.




        


        
        
    


    



    
Медицинский отказ от ответственности

    

        This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.
    

    

        Data sources:
        ChEMBL,
        PubChem,
        DailyMed.