Chloroprocaine Hydrochloride

CHEMBL944 Phase 4 Одобрено Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
307.2 g/mol
LogP
Phase
4

The hydrochloride salt formulation of chloroprocaine is the clinical preparation used for epidural and infiltration anesthesia. It shares the rapid onset and short duration of action of the parent compound due to fast ester hydrolysis. It is favored in labor analgesia and ambulatory surgical settings.

Молекулярная масса

307,2100 g/mol

TPSA

55,60 Ų

Терапевтические области

Механизм действия

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Механизм

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

2D Структура

SVG PNG

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SMILES

CCN(CC)CCOC(=O)c1ccc(N)cc1Cl.Cl

InChI

InChI=1S/C13H19ClN2O2.ClH/c1-3-16(4-2)7-8-18-13(17)11-6-5-10(15)9-12(11)14;/h5-6,9H,3-4,7-8,15H2,1-2H3;1H

Molecular Formula

C13H20Cl2N2O2

HBD / HBA

2 / 4

Вращаемые Связи

7

Тяжёлые Атомы

19

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Часто задаваемые вопросы

The hydrochloride salt formulation of chloroprocaine is the clinical preparation used for epidural and infiltration anesthesia. It shares the rapid onset and short duration of action of the parent compound due to fast ester hydrolysis. It is favored in labor analgesia and ambulatory surgical settings.

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Yes, Chloroprocaine Hydrochloride is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL944. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 441348. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

Медицинский отказ от ответственности

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.