Zaleplon

CHEMBL1521 Phase 4 Одобрено Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
305.3 g/mol
LogP
1.0
Phase
4

This non-benzodiazepine sleep aid is prescribed for the short-term treatment of insomnia, specifically to help people fall asleep faster. It works by binding to GABA receptors in the brain in a way similar to benzodiazepines, producing a calming, sleep-inducing effect. Its very short duration of action means it is less likely to cause next-morning grogginess, but complex sleep behaviors (such as sleepwalking) have been reported.

Молекулярная масса

305,3300 g/mol

LogP

1,00

TPSA

74,30 Ų

Правило пяти Липинского

Соответствует

Терапевтические области

Pharmacokinetics (PK)

Pharmacodynamics (PD)

2D Структура

SVG PNG

Cite this structure


                        

Embed this structure


                        

SMILES

CCN(C(C)=O)c1cccc(-c2ccnc3c(C#N)cnn23)c1

InChI

InChI=1S/C17H15N5O/c1-3-21(12(2)23)15-6-4-5-13(9-15)16-7-8-19-17-14(10-18)11-20-22(16)17/h4-9,11H,3H2,1-2H3

Molecular Formula

C17H15N5O

HBD / HBA

- / 4

Вращаемые Связи

3

Тяжёлые Атомы

23

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Часто задаваемые вопросы

This non-benzodiazepine sleep aid is prescribed for the short-term treatment of insomnia, specifically to help people fall asleep faster. It works by binding to GABA receptors in the brain in a way similar to benzodiazepines, producing a calming, sleep-inducing effect. Its very short duration of action means it is less likely to cause next-morning grogginess, but complex sleep behaviors (such as sleepwalking) have been reported.

Yes, Zaleplon is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1521. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 5719. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

Медицинский отказ от ответственности

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.