PPARG (Peroxisome Proliferator-Activated Receptor Gamma)
PPARG
Nuclear receptor regulating glucose and lipid metabolism, adipocyte differentiation.
Функция
Thiazolidinediones (pioglitazone) activate PPARG to improve insulin sensitivity.
Препараты, действующие на данную мишень
| Препарат | Действие | Первичный |
|---|---|---|
| Methylprednisolone | Agonist | Да |
| Insulin Glargine | Agonist | Да |
| Liraglutide | Agonist | Да |
| Semaglutide | Agonist | Да |
| Tirzepatide | Agonist | Да |
| Prednisone | Agonist | Да |
| Dexamethasone | Agonist | Да |
| Levothyroxine | Agonist | Да |
| Spironolactone | Antagonist | Да |
| Tamoxifen | Antagonist | Да |
| Sitagliptin | Inhibitor | Да |
| Finasteride | Inhibitor | Да |
| Empagliflozin | Inhibitor | Да |
| Metformin | Other | Да |
| Montelukast | Other | — |