Brimonidine Tartrate

CHEMBL1200389 Phase 4 ได้รับการอนุมัติ Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
442.2 g/mol
LogP
Phase
4

The tartrate salt of brimonidine, commonly formulated as ophthalmic drops to reduce elevated eye pressure in glaucoma. It works by decreasing fluid production inside the eye and enhancing uveoscleral outflow. It should be used with caution in young children due to the risk of central nervous system depression.

น้ำหนักโมเลกุล

442.2200 g/mol

TPSA

177.00 Ų

ด้านการรักษา

กลไกการออกฤทธิ์

Absorbs, reflects, or scatters ultraviolet radiation before it reaches the skin, protecting against UV-induced DNA damage and sunburn.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

กลไก

Absorbs, reflects, or scatters ultraviolet radiation before it reaches the skin, protecting against UV-induced DNA damage and sunburn.

โครงสร้าง 2 มิติ

SVG PNG

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SMILES

Brc1c(NC2=NCCN2)ccc2nccnc12.O=C(O)[C@H](O)[C@@H](O)C(=O)O

InChI

InChI=1S/C11H10BrN5.C4H6O6/c12-9-7(17-11-15-5-6-16-11)1-2-8-10(9)14-4-3-13-8;5-1(3(7)8)2(6)4(9)10/h1-4H,5-6H2,(H2,15,16,17);1-2,5-6H,(H,7,8)(H,9,10)/t;1-,2-/m.1/s1

Molecular Formula

C15H16BrN5O6

HBD / HBA

6 / 9

พันธะที่หมุนได้

5

อะตอมหนัก

27

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

คำถามที่พบบ่อย

The tartrate salt of brimonidine, commonly formulated as ophthalmic drops to reduce elevated eye pressure in glaucoma. It works by decreasing fluid production inside the eye and enhancing uveoscleral outflow. It should be used with caution in young children due to the risk of central nervous system depression.

Absorbs, reflects, or scatters ultraviolet radiation before it reaches the skin, protecting against UV-induced DNA damage and sunburn.

Yes, Brimonidine Tartrate is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1200389. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 54405. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

ข้อจำกัดความรับผิดชอบทางการแพทย์

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.