Eslicarbazepine Acetate

CHEMBL87992 Phase 4 ได้รับการอนุมัติ Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
296.3 g/mol
LogP
2.0
Phase
4

This anticonvulsant is converted in the body to eslicarbazepine, which blocks sodium channels in neurons to reduce abnormal electrical activity in the brain. It is used as an add-on treatment for partial-onset seizures.

น้ำหนักโมเลกุล

296.3200 g/mol

LogP

2.00

TPSA

72.60 Ų

Lipinski RO5

ผ่าน

ด้านการรักษา

กลไกการออกฤทธิ์

Selectively blocks angiotensin II type 1 (AT1) receptors, preventing the vasoconstrictive and aldosterone-secreting effects of angiotensin II. This results in vasodilation, reduced sodium retention, and decreased blood pressure.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

กลไก

Selectively blocks angiotensin II type 1 (AT1) receptors, preventing the vasoconstrictive and aldosterone-secreting effects of angiotensin II. This results in vasodilation, reduced sodium retention, and decreased blood pressure.

โครงสร้าง 2 มิติ

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SMILES

CC(=O)O[C@H]1Cc2ccccc2N(C(N)=O)c2ccccc21

InChI

InChI=1S/C17H16N2O3/c1-11(20)22-16-10-12-6-2-4-8-14(12)19(17(18)21)15-9-5-3-7-13(15)16/h2-9,16H,10H2,1H3,(H2,18,21)/t16-/m0/s1

Molecular Formula

C17H16N2O3

HBD / HBA

1 / 3

พันธะที่หมุนได้

2

อะตอมหนัก

22

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

คำถามที่พบบ่อย

This anticonvulsant is converted in the body to eslicarbazepine, which blocks sodium channels in neurons to reduce abnormal electrical activity in the brain. It is used as an add-on treatment for partial-onset seizures.

Selectively blocks angiotensin II type 1 (AT1) receptors, preventing the vasoconstrictive and aldosterone-secreting effects of angiotensin II. This results in vasodilation, reduced sodium retention, and decreased blood pressure.

Yes, Eslicarbazepine Acetate is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL87992. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 179344. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

ข้อจำกัดความรับผิดชอบทางการแพทย์

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.