Anileridine

CHEMBL1201347 Phase 4 Onaylandı Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
352.5 g/mol
LogP
3.7
Phase
4

An opioid analgesic that binds to mu-opioid receptors in the brain and spinal cord to relieve moderate to severe pain. Like other opioids, it carries risks of respiratory depression, dependence, and tolerance.

Moleküler Ağırlık

352,5000 g/mol

LogP

3,70

TPSA

55,60 Ų

Lipinski RO5

Geçer

Etki Mekanizması

Binds to mu (μ), kappa (κ), and/or delta (δ) opioid receptors in the central and peripheral nervous system, mimicking endogenous endorphins. Activation of these G-protein-coupled receptors inhibits pain signal transmission and modulates the emotional response to pain.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Mekanizma

Binds to mu (μ), kappa (κ), and/or delta (δ) opioid receptors in the central and peripheral nervous system, mimicking endogenous endorphins. Activation of these G-protein-coupled receptors inhibits pain signal transmission …

2D Yapı

SVG PNG

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SMILES

CCOC(=O)C1(c2ccccc2)CCN(CCc2ccc(N)cc2)CC1

InChI

InChI=1S/C22H28N2O2/c1-2-26-21(25)22(19-6-4-3-5-7-19)13-16-24(17-14-22)15-12-18-8-10-20(23)11-9-18/h3-11H,2,12-17,23H2,1H3

Molecular Formula

C22H28N2O2

HBD / HBA

1 / 4

Döndürülebilir Bağlar

7

Ağır Atomlar

26

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Sıkça Sorulan Sorular

An opioid analgesic that binds to mu-opioid receptors in the brain and spinal cord to relieve moderate to severe pain. Like other opioids, it carries risks of respiratory depression, dependence, and tolerance.

Binds to mu (μ), kappa (κ), and/or delta (δ) opioid receptors in the central and peripheral nervous system, mimicking endogenous endorphins. Activation of these G-protein-coupled receptors inhibits pain signal transmission and modulates the emotional response to pain.

Yes, Anileridine is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1201347. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 8944. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

Tıbbi Sorumluluk Reddi

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.