Dyclonine

CHEMBL1201217 Phase 4 Onaylandı Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
289.4 g/mol
LogP
3.6
Phase
4

A local anesthetic used topically to numb mucous membranes in the mouth and throat. It is commonly found in throat lozenges and sprays to relieve pain from sore throats and mouth sores.

Moleküler Ağırlık

289,4000 g/mol

LogP

3,60

TPSA

29,50 Ų

Lipinski RO5

Geçer

Etki Mekanizması

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Mekanizma

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

2D Yapı

SVG PNG

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SMILES

CCCCOc1ccc(C(=O)CCN2CCCCC2)cc1

InChI

InChI=1S/C18H27NO2/c1-2-3-15-21-17-9-7-16(8-10-17)18(20)11-14-19-12-5-4-6-13-19/h7-10H,2-6,11-15H2,1H3

Molecular Formula

C18H27NO2

HBD / HBA

- / 3

Döndürülebilir Bağlar

8

Ağır Atomlar

21

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Sıkça Sorulan Sorular

A local anesthetic used topically to numb mucous membranes in the mouth and throat. It is commonly found in throat lozenges and sprays to relieve pain from sore throats and mouth sores.

Blocks voltage-gated sodium channels in nerve cell membranes, preventing the generation and conduction of nerve impulses. This produces reversible loss of sensation in the area of application.

Yes, Dyclonine is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1201217. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 3180. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

Tıbbi Sorumluluk Reddi

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.