Isoetharine

CHEMBL1201213 Phase 4 Onaylandı Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
239.3 g/mol
LogP
1.7
Phase
4

This adrenergic bronchodilator was used to relieve bronchospasm in asthma and COPD by stimulating beta-2 receptors in the lungs to relax airway smooth muscle. It has a relatively short duration of action compared to newer beta-agonists. It has largely been superseded by more selective and longer-lasting bronchodilators.

Moleküler Ağırlık

239,3100 g/mol

LogP

1,70

TPSA

72,70 Ų

Lipinski RO5

Geçer

Etki Mekanizması

Activates beta-2 adrenergic receptors on bronchial smooth muscle, stimulating adenylyl cyclase and increasing intracellular cAMP. This relaxes airway smooth muscle and produces bronchodilation.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Mekanizma

Activates beta-2 adrenergic receptors on bronchial smooth muscle, stimulating adenylyl cyclase and increasing intracellular cAMP. This relaxes airway smooth muscle and produces bronchodilation.

2D Yapı

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SMILES

CCC(NC(C)C)C(O)c1ccc(O)c(O)c1

InChI

InChI=1S/C13H21NO3/c1-4-10(14-8(2)3)13(17)9-5-6-11(15)12(16)7-9/h5-8,10,13-17H,4H2,1-3H3

Molecular Formula

C13H21NO3

HBD / HBA

4 / 4

Döndürülebilir Bağlar

5

Ağır Atomlar

17

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Sıkça Sorulan Sorular

This adrenergic bronchodilator was used to relieve bronchospasm in asthma and COPD by stimulating beta-2 receptors in the lungs to relax airway smooth muscle. It has a relatively short duration of action compared to newer beta-agonists. It has largely been superseded by more selective and longer-lasting bronchodilators.

Activates beta-2 adrenergic receptors on bronchial smooth muscle, stimulating adenylyl cyclase and increasing intracellular cAMP. This relaxes airway smooth muscle and produces bronchodilation.

Yes, Isoetharine is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

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References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1201213. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 3762. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

Tıbbi Sorumluluk Reddi

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.