Raltegravir Potassium

CHEMBL518520 Phase 4 Onaylandı Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
482.5 g/mol
LogP
Phase
4

The potassium salt formulation of raltegravir used in combination with other antiretroviral drugs to suppress HIV replication and maintain immune function. It is well-tolerated and has a favorable drug interaction profile compared to some older HIV medications.

Moleküler Ağırlık

482,5000 g/mol

TPSA

153,00 Ų

Terapötik Alanlar

Etki Mekanizması

Inhibits viral integrase, preventing the insertion of viral DNA into the host cell genome and blocking viral replication.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Mekanizma

Inhibits viral integrase, preventing the insertion of viral DNA into the host cell genome and blocking viral replication.

2D Yapı

SVG PNG

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SMILES

Cc1nnc(C(=O)NC(C)(C)c2nc(C(=O)NCc3ccc(F)cc3)c([O-])c(=O)n2C)o1.[K+]

InChI

InChI=1S/C20H21FN6O5.K/c1-10-25-26-17(32-10)16(30)24-20(2,3)19-23-13(14(28)18(31)27(19)4)15(29)22-9-11-5-7-12(21)8-6-11;/h5-8,28H,9H2,1-4H3,(H,22,29)(H,24,30);/q;+1/p-1

Molecular Formula

C20H20FKN6O5

HBD / HBA

2 / 9

Döndürülebilir Bağlar

6

Ağır Atomlar

33

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Sıkça Sorulan Sorular

The potassium salt formulation of raltegravir used in combination with other antiretroviral drugs to suppress HIV replication and maintain immune function. It is well-tolerated and has a favorable drug interaction profile compared to some older HIV medications.

Inhibits viral integrase, preventing the insertion of viral DNA into the host cell genome and blocking viral replication.

Yes, Raltegravir Potassium is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL518520. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 23668479. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

Tıbbi Sorumluluk Reddi

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.