Rivastigmine Tartrate

CHEMBL1201092 Phase 4 Onaylandı Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
400.4 g/mol
LogP
Phase
4

The tartrate salt formulation of rivastigmine used to improve cognitive symptoms in Alzheimer's disease dementia by maintaining higher levels of the neurotransmitter acetylcholine. It helps with memory, thinking, and daily functioning in people with mild to moderate Alzheimer's.

Moleküler Ağırlık

400,4000 g/mol

TPSA

148,00 Ų

Terapötik Alanlar

Etki Mekanizması

Inhibits acetylcholinesterase, the enzyme that hydrolyzes acetylcholine in the synaptic cleft. This increases acetylcholine availability at cholinergic synapses, enhancing cholinergic neurotransmission.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Mekanizma

Inhibits acetylcholinesterase, the enzyme that hydrolyzes acetylcholine in the synaptic cleft. This increases acetylcholine availability at cholinergic synapses, enhancing cholinergic neurotransmission.

2D Yapı

SVG PNG

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SMILES

CCN(C)C(=O)Oc1cccc([C@H](C)N(C)C)c1.O=C(O)[C@H](O)[C@@H](O)C(=O)O

InChI

InChI=1S/C14H22N2O2.C4H6O6/c1-6-16(5)14(17)18-13-9-7-8-12(10-13)11(2)15(3)4;5-1(3(7)8)2(6)4(9)10/h7-11H,6H2,1-5H3;1-2,5-6H,(H,7,8)(H,9,10)/t11-;1-,2-/m01/s1

Molecular Formula

C18H28N2O8

HBD / HBA

4 / 9

Döndürülebilir Bağlar

8

Ağır Atomlar

28

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Sıkça Sorulan Sorular

The tartrate salt formulation of rivastigmine used to improve cognitive symptoms in Alzheimer's disease dementia by maintaining higher levels of the neurotransmitter acetylcholine. It helps with memory, thinking, and daily functioning in people with mild to moderate Alzheimer's.

Inhibits acetylcholinesterase, the enzyme that hydrolyzes acetylcholine in the synaptic cleft. This increases acetylcholine availability at cholinergic synapses, enhancing cholinergic neurotransmission.

Yes, Rivastigmine Tartrate is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1201092. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 6918078. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

Tıbbi Sorumluluk Reddi

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.