Tocainide Hydrochloride

CHEMBL1200773 Phase 4 已批准 Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
228.7 g/mol
LogP
Phase
4

Tocainide hydrochloride is the hydrochloride salt form of tocainide, an oral class Ib antiarrhythmic agent that blocks voltage-gated sodium channels in ventricular myocardium. See tocainide for complete pharmacological details. This salt formulation was used in oral preparations prior to market withdrawal due to severe hematological and pulmonary toxicity.

分子量

228.7200 g/mol

TPSA

55.10 Ų

Pharmacokinetics (PK)

Pharmacodynamics (PD)

二维结构

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SMILES

Cc1cccc(C)c1NC(=O)C(C)N.Cl

InChI

InChI=1S/C11H16N2O.ClH/c1-7-5-4-6-8(2)10(7)13-11(14)9(3)12;/h4-6,9H,12H2,1-3H3,(H,13,14);1H

Molecular Formula

C11H17ClN2O

HBD / HBA

3 / 2

可旋转键数

2

重原子数

15

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

常见问题

Tocainide hydrochloride is the hydrochloride salt form of tocainide, an oral class Ib antiarrhythmic agent that blocks voltage-gated sodium channels in ventricular myocardium. See tocainide for complete pharmacological details. This salt formulation was used in oral preparations prior to market withdrawal due to severe hematological and pulmonary toxicity.

Yes, Tocainide Hydrochloride is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1200773. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 108173. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

医疗免责声明

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.