Echothiophate

CHEMBL1201341 Phase 4 معتمد Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
256.3 g/mol
LogP
1.0
Phase
4

An organophosphate cholinesterase inhibitor used as an eye drop to treat glaucoma and certain types of strabismus (crossed eyes). It reduces intraocular pressure by promoting the drainage of fluid from the eye.

الوزن الجزيئي

256,3300 g/mol

LogP

1,00

TPSA

60,80 Ų

قاعدة ليبينسكي للخمسة

ناجح

آلية العمل

Inhibits acetylcholinesterase, the enzyme that hydrolyzes acetylcholine in the synaptic cleft. This increases acetylcholine availability at cholinergic synapses, enhancing cholinergic neurotransmission.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

الآلية

Inhibits acetylcholinesterase, the enzyme that hydrolyzes acetylcholine in the synaptic cleft. This increases acetylcholine availability at cholinergic synapses, enhancing cholinergic neurotransmission.

البنية ثنائية الأبعاد

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SMILES

CCOP(=O)(OCC)SCC[N+](C)(C)C

InChI

InChI=1S/C9H23NO3PS/c1-6-12-14(11,13-7-2)15-9-8-10(3,4)5/h6-9H2,1-5H3/q+1

Molecular Formula

C9H23NO3PS+

HBD / HBA

- / 4

الروابط القابلة للدوران

8

الذرات الثقيلة

15

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

الأسئلة الشائعة

An organophosphate cholinesterase inhibitor used as an eye drop to treat glaucoma and certain types of strabismus (crossed eyes). It reduces intraocular pressure by promoting the drainage of fluid from the eye.

Inhibits acetylcholinesterase, the enzyme that hydrolyzes acetylcholine in the synaptic cleft. This increases acetylcholine availability at cholinergic synapses, enhancing cholinergic neurotransmission.

Yes, Echothiophate is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1201341. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 10548. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

إخلاء المسؤولية الطبية

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.