Quinupristin

CHEMBL1200649 Phase 4 معتمد Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
1022.2 g/mol
LogP
4.2
Phase
4

An antibiotic used in combination with dalfopristin to treat serious infections caused by certain gram-positive bacteria, including vancomycin-resistant strains. It works by blocking bacterial protein synthesis at two different points, making it difficult for bacteria to develop resistance.

الوزن الجزيئي

1022,2000 g/mol

LogP

4,20

TPSA

257,00 Ų

قاعدة ليبينسكي للخمسة

راسب

Pharmacokinetics (PK)

Pharmacodynamics (PD)

البنية ثنائية الأبعاد

SVG PNG

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SMILES

CC[C@H]1NC(=O)[C@@H](NC(=O)c2ncccc2O)[C@@H](C)OC(=O)[C@H](c2ccccc2)NC(=O)[C@@H]2CC(=O)[C@H](CS[C@@H]3CN4CCC3CC4)CN2C(=O)[C@H](Cc2ccc(N(C)C)cc2)N(C)C(=O)[C@@H]2CCCN2C1=O

InChI

InChI=1S/C53H67N9O10S/c1-6-37-50(68)61-23-11-14-38(61)51(69)59(5)40(26-32-16-18-36(19-17-32)58(3)4)52(70)62-28-35(30-73-43-29-60-24-20-33(43)21-25-60)42(64)27-39(62)47(65)57-45(34-12-8-7-9-13-34)53(71)72-31(2)44(48(66)55-37)56-49(67)46-41(63)15-10-22-54-46/h7-10,12-13,15-19,22,31,33,35,37-40,43-45,63H,6,11,14,20-21,23-30H2,1-5H3,(H,55,66)(H,56,67)(H,57,65)/t31-,35+,37-,38+,39+,40+,43-,44+,45+/m1/s1

Molecular Formula

C53H67N9O10S

HBD / HBA

4 / 14

الروابط القابلة للدوران

10

الذرات الثقيلة

73

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

الأسئلة الشائعة

An antibiotic used in combination with dalfopristin to treat serious infections caused by certain gram-positive bacteria, including vancomycin-resistant strains. It works by blocking bacterial protein synthesis at two different points, making it difficult for bacteria to develop resistance.

Yes, Quinupristin is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1200649. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 5388937. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

إخلاء المسؤولية الطبية

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.