Methoxamine
A selective alpha-1 adrenergic agonist vasopressor used to raise blood pressure, particularly to treat hypotension during spinal anesthesia. It is administered by injection in clinical settings.
Molecular Weight
211.2600 g/mol
LogP
0.50
TPSA
64.70 Ų
Lipinski RO5
Pass
Pharmacokinetics (PK)
Pharmacodynamics (PD)
2D Structure
Cite this structure
Embed this structure
SMILES
COc1ccc(OC)c(C(O)C(C)N)c1
InChI
InChI=1S/C11H17NO3/c1-7(12)11(13)9-6-8(14-2)4-5-10(9)15-3/h4-7,11,13H,12H2,1-3H3
Molecular Formula
C11H17NO3
HBD / HBA
2 / 4
Rotatable Bonds
4
Heavy Atoms
15
No targets recorded
Target interaction data is not yet available for this drug.
No interactions recorded
Drug interaction data is not yet available for this compound.
No side effects recorded
Side effect data is not yet available for this drug.
Frequently Asked Questions
A selective alpha-1 adrenergic agonist vasopressor used to raise blood pressure, particularly to treat hypotension during spinal anesthesia. It is administered by injection in clinical settings.
Yes, Methoxamine is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.
References & Data Sources
- ChEMBL — European Bioinformatics Institute (EBI). CHEMBL524. Open-access bioactivity database.
- PubChem — National Center for Biotechnology Information (NCBI). CID 6082. Chemical information database.
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.
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