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Tapentadol

CHEMBL1201776 Phase 4 Aprobado Small molecule
Half-Life
—
Bioavailability
—
Protein Binding
—
Molecular Weight
221.3 g/mol
LogP
3.5
Phase
4

This is a prescription opioid pain reliever used to manage moderate to severe pain, including long-term (chronic) pain in adults. It works both by binding to opioid receptors and by blocking the reuptake of norepinephrine, a brain chemical involved in pain signaling. Like all opioids, it carries a risk of dependence and should be used only as directed by a doctor.

Peso molecular

221,3400 g/mol

LogP

3,50

TPSA

23,50 Ų

Regla de cinco de Lipinski

Cumple

Áreas terapéuticas

Artritis reumatoide Cáncer colorrectal Cáncer de mama Cáncer de ovario Cáncer de páncreas Cáncer de próstata Cáncer de pulmón de células no pequeñas Cáncer de tiroides Cáncer de vejiga Dolor crónico Manejo del dolor

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Estructura 2D

SVG PNG

Cite this structure


                        

                            
                            
                        

                    

                


                
                

                    

                    

                        
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SMILES

                    
CC[C@@H](c1cccc(O)c1)[C@@H](C)CN(C)C

                

                

                
                

                    
InChI

                    
InChI=1S/C14H23NO/c1-5-14(11(2)10-15(3)4)12-7-6-8-13(16)9-12/h6-9,11,14,16H,5,10H2,1-4H3/t11-,14+/m0/s1

                

                

                

                    
                    

                        
Molecular Formula

                        
C14H23NO

                    

                    
                    

                        
HBD / HBA

                        
1 / 2

                    

                    
                    

                        
Enlaces Rotables

                        
5

                    

                    
                    
                    

                        
Átomos Pesados

                        
16

                    

                    
                

            


            
            

                
                


    
    
        
    
    
    
No targets recorded

    
    
Target interaction data is not yet available for this drug.

    



                
            


            
            

                
                


    
    
        
    
    
    
No interactions recorded

    
    
Drug interaction data is not yet available for this compound.

    



                
            


            
            

                
                


    
    
        
    
    
    
No side effects recorded

    
    
Side effect data is not yet available for this drug.

    



                
            


            
            
            

                
Preguntas frecuentes

                

                    
                    

                        
                        

                            
This is a prescription opioid pain reliever used to manage moderate to severe pain, including long-term (chronic) pain in adults. It works both by binding to opioid receptors and by blocking the reuptake of norepinephrine, a brain chemical involved in pain signaling. Like all opioids, it carries a risk of dependence and should be used only as directed by a doctor.

                        

                    

                    

                    

                    

                    

                    

                        
                        

                            
Yes, Tapentadol is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

                        

                    

                

            

            

            
            

            
            

            
            
{# References & Data Sources section for drug detail pages.
   Renders standard pharmacological database links plus the drug's data_sources field. #}


    
References & Data Sources

    
    
        
        
  • 
            
            
                ChEMBL — European Bioinformatics Institute (EBI).
                CHEMBL1201776.
                Open-access bioactivity database.
            
        
    • 
        
        
        
  • 
            
            
                PubChem — National Center for Biotechnology Information (NCBI).
                CID 9838022.
                Chemical information database.
            
        
    • 
        
        
        
        
    

    
Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.




        


        
        
    


    



    
Aviso médico

    

        This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.
    

    

        Data sources:
        ChEMBL,
        PubChem,
        DailyMed.