Sufentanil

CHEMBL658 Phase 4 Approuvé Small molecule

Half-Life

—

Bioavailability

—

Protein Binding

—

Molecular Weight

386.6 g/mol

LogP

4.0

Phase

4

A potent synthetic opioid approximately 5 to 10 times stronger than fentanyl, used in carefully controlled anesthetic and intensive care settings to provide powerful pain relief and sedation. A sublingual microtablet formulation has also been developed for managing moderate to severe acute pain in supervised healthcare settings.

Masse moléculaire

386,6000 g/mol

LogP

4,00

TPSA

61,00 Å²

Règle des 5 de Lipinski

Conforme

Aires thérapeutiques

Ovarian Cancer Pancreatic Cancer Bladder Cancer Thyroid Cancer Cardiovascular Disease Pain Management Non-Small Cell Lung Cancer Parkinson's Disease Generalized Anxiety Disorder Melanoma Oncology Inflammatory Bowel Disease Chronic Kidney Disease Stroke Obesity Hypertension Breast Cancer Chronic Pain Atrial Fibrillation Prostate Cancer Colorectal Cancer

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Structure 2D

SVG PNG

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SMILES

CCC(=O)N(c1ccccc1)C1(COC)CCN(CCc2cccs2)CC1

InChI

InChI=1S/C22H30N2O2S/c1-3-21(25)24(19-8-5-4-6-9-19)22(18-26-2)12-15-23(16-13-22)14-11-20-10-7-17-27-20/h4-10,17H,3,11-16,18H2,1-2H3

Molecular Formula

C22H30N2O2S

HBD / HBA

- / 4

Liaisons Rotatives

8

Atomes Lourds

27

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Foire aux questions

A potent synthetic opioid approximately 5 to 10 times stronger than fentanyl, used in carefully controlled anesthetic and intensive care settings to provide powerful pain relief and sedation. A sublingual microtablet formulation has also been developed for managing moderate to severe acute pain in supervised healthcare settings.

Yes, Sufentanil is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

ChEMBL — European Bioinformatics Institute (EBI). CHEMBL658. Open-access bioactivity database.
PubChem — National Center for Biotechnology Information (NCBI). CID 41693. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

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Structure

Données Clés

Formule: C22H30N2O2S
Synonymes: 2

Liens externes

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Avertissement médical

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.