Tapentadol

CHEMBL1201776 Phase 4 Approuvé Small molecule

Half-Life

—

Bioavailability

—

Protein Binding

—

Molecular Weight

221.3 g/mol

LogP

3.5

Phase

4

This is a prescription opioid pain reliever used to manage moderate to severe pain, including long-term (chronic) pain in adults. It works both by binding to opioid receptors and by blocking the reuptake of norepinephrine, a brain chemical involved in pain signaling. Like all opioids, it carries a risk of dependence and should be used only as directed by a doctor.

Masse moléculaire

221,3400 g/mol

LogP

3,50

TPSA

23,50 Å²

Règle des 5 de Lipinski

Conforme

Aires thérapeutiques

Ovarian Cancer Pancreatic Cancer Bladder Cancer Thyroid Cancer Pain Management Non-Small Cell Lung Cancer Rheumatoid Arthritis Breast Cancer Chronic Pain Prostate Cancer Colorectal Cancer

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Structure 2D

SVG PNG

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SMILES

CC[C@@H](c1cccc(O)c1)[C@@H](C)CN(C)C

InChI

InChI=1S/C14H23NO/c1-5-14(11(2)10-15(3)4)12-7-6-8-13(16)9-12/h6-9,11,14,16H,5,10H2,1-4H3/t11-,14+/m0/s1

Molecular Formula

C14H23NO

HBD / HBA

1 / 2

Liaisons Rotatives

5

Atomes Lourds

16

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Foire aux questions

This is a prescription opioid pain reliever used to manage moderate to severe pain, including long-term (chronic) pain in adults. It works both by binding to opioid receptors and by blocking the reuptake of norepinephrine, a brain chemical involved in pain signaling. Like all opioids, it carries a risk of dependence and should be used only as directed by a doctor.

Yes, Tapentadol is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1201776. Open-access bioactivity database.
PubChem — National Center for Biotechnology Information (NCBI). CID 9838022. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-28.

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Structure

Données Clés

Formule: C14H23NO
Synonymes: 2

Liens externes

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Avertissement médical

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.