Agonist

Pharmacodynamics

A substance that binds to a receptor and activates it to produce a biological response. Full agonists produce maximal response; partial agonists produce submaximal response even at full receptor occupancy.

Contoh

  • Morphine (full mu-opioid agonist)
  • Buprenorphine (partial agonist)
  • Albuterol (beta-2 agonist)

Tahukah Anda?

A substance that binds to a receptor and activates it to produce a biological response. Full agonists produce maximal response; partial agonists produce submaximal response even at full receptor occupancy.