Echothiophate

CHEMBL1201341 Phase 4 承認済み Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
256.3 g/mol
LogP
1.0
Phase
4

An organophosphate cholinesterase inhibitor used as an eye drop to treat glaucoma and certain types of strabismus (crossed eyes). It reduces intraocular pressure by promoting the drainage of fluid from the eye.

分子量

256.3300 g/mol

LogP

1.00

TPSA

60.80 Ų

リピンスキーの五則

適合

作用機序

Inhibits acetylcholinesterase, the enzyme that hydrolyzes acetylcholine in the synaptic cleft. This increases acetylcholine availability at cholinergic synapses, enhancing cholinergic neurotransmission.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

機序

Inhibits acetylcholinesterase, the enzyme that hydrolyzes acetylcholine in the synaptic cleft. This increases acetylcholine availability at cholinergic synapses, enhancing cholinergic neurotransmission.

2D構造

SVG PNG

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SMILES

CCOP(=O)(OCC)SCC[N+](C)(C)C

InChI

InChI=1S/C9H23NO3PS/c1-6-12-14(11,13-7-2)15-9-8-10(3,4)5/h6-9H2,1-5H3/q+1

Molecular Formula

C9H23NO3PS+

HBD / HBA

- / 4

回転可能結合数

8

重原子数

15

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

よくある質問

An organophosphate cholinesterase inhibitor used as an eye drop to treat glaucoma and certain types of strabismus (crossed eyes). It reduces intraocular pressure by promoting the drainage of fluid from the eye.

Inhibits acetylcholinesterase, the enzyme that hydrolyzes acetylcholine in the synaptic cleft. This increases acetylcholine availability at cholinergic synapses, enhancing cholinergic neurotransmission.

Yes, Echothiophate is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1201341. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 10548. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

医学的免責事項

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.