Cyclopentolate Hydrochloride

CHEMBL1200473 Phase 4 Aprovado Small molecule
Half-Life
Bioavailability
Protein Binding
Molecular Weight
327.8 g/mol
LogP
Phase
4

The hydrochloride salt formulation of cyclopentolate, a mydriatic and cycloplegic agent used as eye drops to dilate the pupil and temporarily paralyze accommodation for eye examinations. It has a faster onset and shorter duration than atropine.

Peso Molecular

327,8000 g/mol

TPSA

49,80 Ų

Áreas Terapêuticas

Mecanismo de Ação

Competitively blocks muscarinic acetylcholine receptors, reducing parasympathetic nervous system activity. Effects include decreased secretions, bronchodilation, and relaxation of smooth muscle.

Pharmacokinetics (PK)

Pharmacodynamics (PD)

Mecanismo

Competitively blocks muscarinic acetylcholine receptors, reducing parasympathetic nervous system activity. Effects include decreased secretions, bronchodilation, and relaxation of smooth muscle.

Estrutura 2D

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SMILES

CN(C)CCOC(=O)C(c1ccccc1)C1(O)CCCC1.Cl

InChI

InChI=1S/C17H25NO3.ClH/c1-18(2)12-13-21-16(19)15(14-8-4-3-5-9-14)17(20)10-6-7-11-17;/h3-5,8-9,15,20H,6-7,10-13H2,1-2H3;1H

Molecular Formula

C17H26ClNO3

HBD / HBA

2 / 4

Ligações Rotacionáveis

7

Átomos Pesados

22

No targets recorded

Target interaction data is not yet available for this drug.

No interactions recorded

Drug interaction data is not yet available for this compound.

No side effects recorded

Side effect data is not yet available for this drug.

Perguntas frequentes

The hydrochloride salt formulation of cyclopentolate, a mydriatic and cycloplegic agent used as eye drops to dilate the pupil and temporarily paralyze accommodation for eye examinations. It has a faster onset and shorter duration than atropine.

Competitively blocks muscarinic acetylcholine receptors, reducing parasympathetic nervous system activity. Effects include decreased secretions, bronchodilation, and relaxation of smooth muscle.

Yes, Cyclopentolate Hydrochloride is an approved drug. It has reached clinical phase 4. It is classified as a Small molecule.

{# References & Data Sources section for drug detail pages. Renders standard pharmacological database links plus the drug's data_sources field. #}

References & Data Sources

  • ChEMBL — European Bioinformatics Institute (EBI). CHEMBL1200473. Open-access bioactivity database.
  • PubChem — National Center for Biotechnology Information (NCBI). CID 22162. Chemical information database.

Data aggregated from publicly available pharmacological databases. Last updated 2026-03-04.

Aviso Médico

This content is for educational and informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before making medication decisions.

Data sources: ChEMBL, PubChem, DailyMed.