Alvos Farmacológicos
Alvos biológicos com os quais os medicamentos interagem.
ABCB1 (P-glycoprotein)
ABCB1
Transporter
ACE (Angiotensin-Converting Enzyme)
ACE
Enzyme
ADRB1 (Beta-1 Adrenergic Receptor)
ADRB1
Receptor
ADRB2 (Beta-2 Adrenergic Receptor)
ADRB2
Receptor
AGTR1 (Angiotensin II Type 1 Receptor)
AGTR1
Receptor
ALK (Anaplastic Lymphoma Kinase)
ALK
Kinase
ATP4A (Proton Pump (H+/K+-ATPase))
ATP4A
Enzyme
BCR-ABL1 (BCR-ABL Fusion Protein)
BCR-ABL1
Kinase
BRAF (BRAF Kinase)
BRAF
Kinase
CDK4/CDK6 (Cyclin-Dependent Kinase 4/6)
CDK4/CDK6
Kinase
CTLA4 (Cytotoxic T-Lymphocyte Antigen 4)
CTLA4
Receptor
CYP2D6 (Cytochrome P450 2D6)
CYP2D6
Enzyme
CYP3A4 (Cytochrome P450 3A4)
CYP3A4
Enzyme
DRD2 (Dopamine D2 Receptor)
DRD2
Receptor
EGFR (Epidermal Growth Factor Receptor)
EGFR
Kinase
F10 (Factor Xa)
F10
Protease
F2 (Thrombin)
F2
Protease
GABRA1 (GABA-A Receptor)
GABRA1
Ion Channel
HMGCR (HMG-CoA Reductase)
HMGCR
Enzyme
HRH1 (Histamine H1 Receptor)
HRH1
Receptor
HRH2 (Histamine H2 Receptor)
HRH2
Receptor
HTR2A (Serotonin 5-HT2A Receptor)
HTR2A
Receptor
IL6 (Interleukin-6)
IL6
Other
KDR (Vascular Endothelial Growth Factor Receptor 2)
KDR
Kinase
MTOR (Mechanistic Target of Rapamycin)
MTOR
Kinase
OPRM1 (Mu-Opioid Receptor)
OPRM1
Receptor
PDCD1 (Programmed Cell Death Protein 1)
PDCD1
Receptor
PDE5A (Phosphodiesterase 5)
PDE5A
Enzyme
PPARG (Peroxisome Proliferator-Activated Receptor Gamma)
PPARG
Nuclear Receptor
PTGS1 (Cyclooxygenase-1)
PTGS1
Enzyme
PTGS2 (Cyclooxygenase-2)
PTGS2
Enzyme
SCN9A (Sodium Channel Nav1.7)
SCN9A
Ion Channel
SIGMAR1 (Sigma-1 Receptor)
SIGMAR1
Receptor
SLC6A4 (Serotonin Transporter)
SLC6A4
Transporter
TNF (Tumor Necrosis Factor Alpha)
TNF
Other
VKORC1 (Vitamin K Epoxide Reductase)
VKORC1
Enzyme