SCN9A (Sodium Channel Nav1.7)
SCN9A
Voltage-gated sodium channel preferentially expressed in nociceptive neurons.
Função
Gain-of-function mutations cause inherited pain disorders. Blocking reduces pain signaling.
Medicamentos que Atuam neste Alvo
| Medicamento | Ação | Primário |
|---|---|---|
| Valproic Acid | Blocker | Sim |
| Topiramate | Blocker | Sim |
| Phenytoin | Blocker | Sim |
| Gabapentin | Blocker | Sim |
| Pregabalin | Blocker | Sim |
| Lamotrigine | Blocker | Sim |
| Carbamazepine | Blocker | Sim |
| Furosemide | Inhibitor | Sim |
| Hydrochlorothiazide | Inhibitor | Sim |