SCN9A (Sodium Channel Nav1.7)
SCN9A
Voltage-gated sodium channel preferentially expressed in nociceptive neurons.
功能
Gain-of-function mutations cause inherited pain disorders. Blocking reduces pain signaling.
作用于该靶点的药物
| 药物 | 作用 | 主要 |
|---|---|---|
| Valproic Acid | Blocker | 是 |
| Topiramate | Blocker | 是 |
| Phenytoin | Blocker | 是 |
| Gabapentin | Blocker | 是 |
| Pregabalin | Blocker | 是 |
| Lamotrigine | Blocker | 是 |
| Carbamazepine | Blocker | 是 |
| Furosemide | Inhibitor | 是 |
| Hydrochlorothiazide | Inhibitor | 是 |