GABRA1 (GABA-A Receptor)
GABRA1
Ligand-gated chloride channel mediating fast inhibitory neurotransmission in the CNS.
功能
Benzodiazepines, barbiturates, and general anesthetics enhance GABA-A receptor function via allosteric modulation.
作用于该靶点的药物
| 药物 | 作用 | 主要 |
|---|---|---|
| Diazepam | Agonist | 是 |
| Alprazolam | Agonist | 是 |
| Zolpidem | Agonist | 是 |
| Memantine | Antagonist | 是 |
| Valproic Acid | Agonist | — |
| Topiramate | Agonist | — |